CAS 129-56-6 SP-600125 is a potent, cell permeable, selective, and reversible inhibitor of c-Jun N-terminal kinase (JNK)

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  • CAS: 129-56-6
  • Formula: C14H8N2O
  • MW: 220.2
  • Appearance: Yellow solid
  • Purity: >98%




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SP600125, SP-600125 is a potent, cell permeable, selective, and reversible inhibitor of c-Jun N-terminal kinase (JNK) (IC50 = 40nM for JNK-1 and JNK-2 and 90nM for JNK-3).
SP600125, SP-600125 exhibits over 300-fold greater selectivity for JNK as compared to ERK1 and p38..

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Product #S-2022
CAS #129-56-6
Chemical Name1,9- Pyrazoloanthrone
AppearanceYellow solid
SolubilitySoluble in DMSO(22 mg/ml) or ethanol (2mg/ml)
Storage Temp-20°C, Store in Tightly Sealed Vial. Protect from Light.

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Certificate of Analysis 1S-2022, H1145B.pdf
Certificate of Analysis 2S-2022, H1145A.pdf
Certificate of Analysis 3S-2022, H1145.pdf
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